Multifaceted biological and computational assessment of aromatic and N-heteroaromatic non-substituted thiosemicarbazones

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Scientific reports - ISSN 2045-2322-16:1 (2026) p. 1-22
Auteur(s)
    Natalia Macijewska, Predrag Ristic, Anoop Kallingal, Mihaela Gulea, Morgan Donnard, Nicolas Girard, An Matheeussen, Natascha Van Pelt, Guy Caljon, Vladimir Dobricic, Jelena Boskovic, Marija Popovic-Nikolic, Katarina Nikolic, Mire Zloh, Vladimir Blagojevic, Tamara Todorovic, Nenad Filipovic

A strategic discovery roadmap towards high-quality leads and drug development candidates for kinetoplastid diseases. Part 1: setting the stage

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The journal of antimicrobial chemotherapy - ISSN 0305-7453-81:5 (2026) p. 1-5
Auteur(s)
    Sarah Hendrickx, Kayhan Ilbeigi, Eli S.J. Thore, Michael G. Bertram, Estefania Calvo-Alvarez, Sener Cintesun, Ana Isabel Olias-Molero, Maria Jesus Corral, Marta Mateo-Barrientos, Jerome Estaquier, Sebastien Pomel, Jose Maria Alunda, Sheraz Gul, Katrien Van Bocxlaer, Frederic Frezard, Joana Tavares, Anabela Cordeiro Da Silva, Maria Paola Costi, Louis Maes, Guy Caljon

A strategic discovery roadmap towards high-quality leads and drug development candidates for kinetoplastid diseases. Part 3: from lead towards a drug development candidate

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The journal of antimicrobial chemotherapy - ISSN 0305-7453-81:6 (2026) p. 1-10
Auteur(s)
    Sarah Hendrickx, Kayhan Ilbeigi, Eli S.J. Thore, Michael G. Bertram, Estefania Calvo-Alvarez, Sener Cintesun, Ana Isabel Olias-Molero, Maria Jesus Corral, Marta Mateo-Barrientos, Jerome Estaquier, Sebastien Pomel, Jose Maria Alunda, Sheraz Gul, Katrien Van Bocxlaer, Frederic Frezard, Joana Tavares, Anabela Cordeiro Da Silva, Maria Paola Costi, Louis Maes, Guy Caljon

A strategic discovery roadmap towards high-quality leads and drug development candidates for kinetoplastid diseases. Part 2: from molecule to confirmed hit

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The journal of antimicrobial chemotherapy - ISSN 0305-7453-81:4 (2026) p. 1-14
Auteur(s)
    Sarah Hendrickx, Kayhan Ilbeigi, Eli S.J. Thore, Michael G. Bertram, Estefania Calvo-Alvarez, Sener Cintesun, Ana Isabel Olias-Molero, Maria Jesus Corral, Marta Mateo-Barrientos, Jerome Estaquier, Sebastien Pomel, Jose Maria Alunda, Sheraz Gul, Katrien Van Bocxlaer, Frederic Frezard, Joana Tavares, Anabela Cordeiro Da Silva, Maria Paola Costi, Louis Maes, Guy Caljon

Bridging antileishmanial drug discovery and cell biology : from mode of action studies to targeting intracellular trafficking

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Antwerp, University of Antwerp, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, Department of Biomedical Sciences, 2026,213 p.