Isolation and characterization of antiplasmodial and antimicrobial compounds from Tetracera alnifolia using a bioassay-guided approach

Source
RSC advances - ISSN 2046-2069-16:12 (2026) p. 10635-10647
Author(s)

Cytotoxicity and antimicrobial activity of GaMF1 analogs

Source
ChemMedChem - ISSN 1860-7179-21:4 (2026) p. 1-17
Author(s)

Collaborative synthesis for neglected diseases through the Open Synthesis Network : structure-activity relationships of arylaminopyrazoles as Chagas disease treatments

Source
ACS Infectious Diseases - ISSN 2373-8227-11:9 (2025) p. 2593-2606
Author(s)
    Zigli Abdulai, Natasha Agbo, Jonathan I. Anderson, Faye Astley, Brian Chan, Owen Atkinson-Evans, Joao L. Avelar, Cristiane Aparecida-Silva, K.D. Bhardwaj, William J. Bowley, Nicholas Breitkreuz, Rosie Canby, Emerald Cartwright, Charles Clifford, Shannon A. Cordell, William J. Donker, Joseph Driscoll, Matthew Grady, Lauren Higginbotham, Devon Hsu, Jamie Hutchinson, Lukas Imberg, Harry F. Jackson, Finan Johns, Emma Jones, Dmitrii V. Kalinin, Ceren Kardesler, Aaron Keal, Libby Keel, Sumin Kim, Phoebe Knight, Justus F. Koedel, Luke Kumeta, Hyejin Lee, Sam Le Roy, Rachelle Maccarone, Maria Mahmud, Matthew Martin, Ignatius Nguyen, Conor J. Nolan, Lucy Noyes, Angela N.W. Ntuwa, Wiktoria Obarska, Owen Oldham, Edna Onyiuke, Jess Otter, Natascha Van Pelt, An Matheeussen, Guy Caljon, Andrew Nortcliffe

Discovery and development of an advanced lead for the treatment of African trypanosomiasis

Source
ACS Infectious Diseases - ISSN 2373-8227-11:1 (2024) p. 131-143
Author(s)

Discovery of a series of macrocycles as potent inhibitors of Leishmania infantum

Source
Journal of medicinal chemistry - ISSN 0022-2623-67:20 (2024) p. 18170-18193
Author(s)
    Federico Riu, Larissa Alena Ruppitsch, Duc Duy Vo, Richard S. Hong, Mohit Tyagi, An Matheeussen, Sarah Hendrickx, Vasanthanathan Poongavanam, Guy Caljon, Ahmad Y. Sheikh, Peter Sjo, Jan Kihlberg